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akaturk Akademik ölçüm

Makale detayı · 2025

Exploring medium and long arm extensions of 1,2,4-triazole derivatives as Candida albicans 14α-demethylase (CYP51) inhibitors

RSC Medicinal Chemistry

YÖKSİS OpenAlex Açık erişim · hybrid SJR Q1 JCR Q2 Atıf 5 Üst %10 Yüzdelik 92.7% FWCI 3.74
Yıl
2025
ISSN
2632-8682
Tür
article

Veri kaynağı ayrımı

  • YÖKSİS YÖKSİS makale kaydı
  • OpenAlex OpenAlex zenginleştirmesi (özet, atıf, konular)

Özet

İngilizce (OpenAlex)

1,2,4-trizole derivatives were designed to study their inhibition of Candida albicans CYP51 (IC 50 ), binding affinity ( K d ) and antifungal profile vs. wild-type and resistant model fungal strains comparable with posaconazole.

Konular

  • Antifungal resistance and susceptibility
  • Peptidase Inhibition and Analysis
  • Biochemical and Molecular Research

Birincil konu Antifungal resistance and susceptibility

Yazarlar

  1. Marwa Alsulaimany
  2. Faizah Binjubair
  3. ESRA TATAR İSTANBUL KENT ÜNİVERSİTESİ
  4. Diane E Kelly
  5. Steven L Kelly
  6. Andrew G Warrilow
  7. Mikhail V Keniya
  8. Brian C Monk
  9. Josie E Parker
  10. Claire Simons